Lead Optimization

BioBlocks, Inc. is highly accomplished at lead optimization. The diverse medicinal chemistry expertise of our management team spans most major therapeutic areas and numerous disease-relevant targets and mechanisms. Our medicinal chemists have developed multiple pre-clinical drug candidates from early leads in a variety of therapeutic areas. This track record enables us to be an effective partner in lead optimization.

Our customers rely on us to bring an insightful collaborative approach to evaluating their initial hits or optimizing their early leads.  BioBlocks’ chemists work with customers to ensure a robust interface with their lead optimization cycles.  We are experienced in applying customers’ SAR and biological testing data to rapidly identify analoging and alternative lead strategies. 

Experience has shown us that our fast cycle time and low-throughput parallel optimization will accelerate lead identification, circumvent roadblocks and reduce project risk.

BioBlocks’ Flex-FTE (Full Time Equivalent) model guarantees that our customer has the chemistry capacity available to successfully overcome the fluctuating demands of projects while meeting project goals, budgets and deadlines.  Our model may include project leadership, consulting on strategy of lead discovery and optimization and integrated chemical information services.  BioBlocks offers highly competitive FTE rates for projects requiring two to six FTEs for six months or longer.

BioBlocks uses secure communications methods and has established procedures to ensure that all confidential information is safeguarded at our San Diego headquarters.

For further information, contact Business Development at 858-558-5900.